{"id":1372,"date":"2021-05-04T08:13:31","date_gmt":"2021-05-04T06:13:31","guid":{"rendered":"https:\/\/portale.unime.it\/modellopersona\/?page_id=31"},"modified":"2025-02-26T12:11:20","modified_gmt":"2025-02-26T11:11:20","slug":"pubblicazioni","status":"publish","type":"page","link":"https:\/\/portale2.unime.it\/desylab\/pubblicazioni\/","title":{"rendered":"PUBBLICAZIONI"},"content":{"rendered":"\t\t<div data-elementor-type=\"wp-page\" data-elementor-id=\"1372\" class=\"elementor elementor-1372\">\n\t\t\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-627a791 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"627a791\" data-element_type=\"section\" data-e-type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-7771bc2\" data-id=\"7771bc2\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap\">\n\t\t\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-66b89f7 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"66b89f7\" data-element_type=\"section\" data-e-type=\"section\" data-settings=\"{&quot;background_background&quot;:&quot;classic&quot;}\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-c8fe409\" data-id=\"c8fe409\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-4687f5d elementor-invisible elementor-widget elementor-widget-heading\" data-id=\"4687f5d\" data-element_type=\"widget\" data-e-type=\"widget\" data-settings=\"{&quot;_animation&quot;:&quot;fadeInDown&quot;}\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h2 class=\"elementor-heading-title elementor-size-default\"><br><br>   PUBBLICAZIONI<br><br><br><\/h2>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-7afe180 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"7afe180\" data-element_type=\"section\" data-e-type=\"section\" data-settings=\"{&quot;background_background&quot;:&quot;classic&quot;}\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-4a87eca elementor-invisible\" data-id=\"4a87eca\" data-element_type=\"column\" data-e-type=\"column\" data-settings=\"{&quot;animation&quot;:&quot;slideInRight&quot;}\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-a127bf2 elementor-widget__width-initial elementor-invisible elementor-widget elementor-widget-heading\" data-id=\"a127bf2\" data-element_type=\"widget\" data-e-type=\"widget\" data-settings=\"{&quot;_animation&quot;:&quot;slideInUp&quot;}\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h4 class=\"elementor-heading-title elementor-size-default\">LE PUBBLICAZIONI\n <\/h4>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-69d13b0 elementor-invisible elementor-widget elementor-widget-heading\" data-id=\"69d13b0\" data-element_type=\"widget\" data-e-type=\"widget\" data-settings=\"{&quot;_animation&quot;:&quot;slideInUp&quot;}\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h4 class=\"elementor-heading-title elementor-size-default\">Il gruppo di ricerca DESY LAB pubblica articoli su riviste scientifiche di interesse internazionale\n <\/h4>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-dafe982 elementor-widget elementor-widget-heading\" data-id=\"dafe982\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h3 class=\"elementor-heading-title elementor-size-default\">Topics: Graphene; Quantum Dot; Biocompatibility; Heavy Metal; Bioaccumulation; Environmental Monitoring; Nitrone; Heterocyclic Compound; Stereoselective Synthesis; Citrus; Flavonoid; Antioxidant Capacity; Antivirus Agent; Nanoparticle; COVID-19; Potassium Channel; Retigabine; Encephalopathy; Transient Receptor Potential Channel; Ankyrin; Sensory Receptor Cell; Human Immunodeficiency Virus 1; Gene Product; RNA<\/h3>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-4c047c8\" data-id=\"4c047c8\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-e46378d elementor-widget elementor-widget-image\" data-id=\"e46378d\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"image.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<img fetchpriority=\"high\" decoding=\"async\" width=\"500\" height=\"500\" src=\"https:\/\/portale2.unime.it\/desylab\/wp-content\/uploads\/sites\/40\/2022\/03\/education-1.png\" class=\"attachment-large size-large wp-image-1277\" alt=\"\" srcset=\"https:\/\/portale2.unime.it\/desylab\/wp-content\/uploads\/sites\/40\/2022\/03\/education-1.png 500w, https:\/\/portale2.unime.it\/desylab\/wp-content\/uploads\/sites\/40\/2022\/03\/education-1-300x300.png 300w, https:\/\/portale2.unime.it\/desylab\/wp-content\/uploads\/sites\/40\/2022\/03\/education-1-150x150.png 150w\" sizes=\"(max-width: 500px) 100vw, 500px\" style=\"width:100%;height:100%;max-width:500px\" \/>\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-7045d58 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"7045d58\" data-element_type=\"section\" data-e-type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-53ba5c4 elementor-invisible\" data-id=\"53ba5c4\" data-element_type=\"column\" data-e-type=\"column\" data-settings=\"{&quot;background_background&quot;:&quot;classic&quot;,&quot;animation&quot;:&quot;fadeInLeft&quot;}\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-fec7e35 elementor-widget elementor-widget-heading\" data-id=\"fec7e35\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h4 class=\"elementor-heading-title elementor-size-default\"><a href=\"https:\/\/portale.unime.it\/modellopersona\/ricerca\/\">RIVISTE<\/a><\/h4>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-4badb3c elementor-view-default elementor-widget elementor-widget-icon\" data-id=\"4badb3c\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"icon.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<div class=\"elementor-icon-wrapper\">\n\t\t\t<div class=\"elementor-icon\">\n\t\t\t<svg aria-hidden=\"true\" class=\"e-font-icon-svg e-fas-book-open\" viewBox=\"0 0 576 512\" xmlns=\"http:\/\/www.w3.org\/2000\/svg\"><path d=\"M542.22 32.05c-54.8 3.11-163.72 14.43-230.96 55.59-4.64 2.84-7.27 7.89-7.27 13.17v363.87c0 11.55 12.63 18.85 23.28 13.49 69.18-34.82 169.23-44.32 218.7-46.92 16.89-.89 30.02-14.43 30.02-30.66V62.75c.01-17.71-15.35-31.74-33.77-30.7zM264.73 87.64C197.5 46.48 88.58 35.17 33.78 32.05 15.36 31.01 0 45.04 0 62.75V400.6c0 16.24 13.13 29.78 30.02 30.66 49.49 2.6 149.59 12.11 218.77 46.95 10.62 5.35 23.21-1.94 23.21-13.46V100.63c0-5.29-2.62-10.14-7.27-12.99z\"><\/path><\/svg>\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-35a161f\" data-id=\"35a161f\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-a9c63f1 elementor-widget elementor-widget-text-editor\" data-id=\"a9c63f1\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t\t\t<p><span style=\"color: #333333\"><span style=\"font-family: tahoma, arial, helvetica, sans-serif;font-size: 10pt\"><strong style=\"background-color: var(--global--color-background)\"><u>RIVISTE<\/u><\/strong><\/span><\/span><\/p><ul style=\"list-style-type: square\"><li><span style=\"font-size: 10pt;color: #000000\">De Gaetano F., Leggio L., Celesti C., Genovese F., Falcone M., <strong>Giofr\u00e8 S.V.,<\/strong> Iraci N., <strong>Iraci N.<\/strong>, Ventura C.A. Study of Host-Guest Interaction and In Vitro Neuroprotective Potential of Cinnamic Acid\/Randomly Methylated \u03b2-Cyclodextrin Inclusion Complex. <em>International Journal of Molecular Sciences<\/em>, <strong>2024<\/strong>, <em>25<\/em> (23), art. no. 12778. DOI: 10.3390\/ijms252312778<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Schiroli D., Voronov A., Pancrazzi F., <strong>Iraci N.<\/strong>, <strong>Giofr\u00e8 S. V.<\/strong>, Macchi B., Stefanizzi V., Mancuso R., Gabriele B., Pio Mazzeo P., Capaldo L., Della Ca&#8217; N. Direct Access to \u03b1,\u03b2-Unsaturated \u03b3-Lactams via Palladium-Catalysed Carbonylation of Propargylic Ureas. <em>Advanced Synthesis and Catalysis<\/em>, <strong>2024<\/strong>, <em>366<\/em>, 1-8. DOI: 10.1002\/adsc.202401183<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">De Gaetano F., Mannino D., Celesti C., Bulzom\u00ed M., <strong>Iraci N.<\/strong>, <strong>Giofr\u00e8 S. V.<\/strong>, Esposito E., Paterniti I., Anna Ventura C. Randomly methylated \u03b2-cyclodextrin improves water \u2013 solubility, cellular protection and mucosa permeability of idebenone. <em>International Journal of Pharmaceutics<\/em>, <strong>2024<\/strong>, <em>665<\/em>, art. no. 124718. DOI: 10.1016\/j.ijpharm.2024.124718<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Di Matteo, F., <strong>Mancuso, F.<\/strong>, Turcio, R., Ciaglia, T., Stagno, C., <strong>Di Chio, C.<\/strong>, Campiglia, P., Bertamino, A., <strong>Giofr\u00e8, S.V.<\/strong>, Ostacolo, C., <strong>Iraci, N. <\/strong>KCNT1 Channel Blockers: A Medicinal Chemistry Perspective, <em>Molecules<\/em>, <strong>2024<\/strong>, 29 (12), art. no. 2940. DOI: 10.3390\/molecules29122940<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Iannazzo, D., <strong>Giofr\u00e8, S.V.<\/strong>, Espro, C., Celesti, C. Graphene-based materials as nanoplatforms for antiviral therapy and prophylaxis. <em>Expert Opinion on Drug Delivery<\/em>, <strong>2024, <\/strong>DOI: 10.1080\/17425247.2024.2364652<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Rossi, A., Stagno, C., Piperno, A., <strong>Iraci, N.<\/strong>, Panseri, S., Montesi, M., Feizi-Dehnayebi, M., Bassi, G., Di Pietro, M.L., Micale, N. Anticancer activity and morphological analysis of Pt (II) complexes: Their DFT approach, docking simulation, and ADME-Tox profiling. <em>Applied Organometallic Chemistry<\/em>, <strong>2024<\/strong>, <em>38<\/em> (5), art. no. e7403. DOI: 10.1002\/aoc.7403<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Sar\u00e0, M., <strong>Giofr\u00e8, S.V.<\/strong>, Abate, S., Trapani, M., Verduci, R., D\u2019Angelo, G., Castriciano, M.A., Romeo, A., Neri, G., Mons\u00f9 Scolaro, L. Absorption and Fluorescence Emission Investigations on Supramolecular Assemblies of Tetrakis-(4-sulfonatophenyl)porphyrin and Graphene Quantum Dots. <em>Molecules<\/em>, <strong>2024<\/strong>, <em>29<\/em> (9), art. no. 2015. DOI: 10.3390\/molecules29092015<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Akbari, Z., Stagno, C., <strong>Iraci, N.<\/strong>, Efferth, T., Omer, E.A., Piperno, A., Montazerozohori, M., Feizi-Dehnayebi, M., Micale, N. Biological evaluation, DFT, MEP, HOMO-LUMO analysis and ensemble docking studies of Zn(II) complexes of bidentate and tetradentate Schiff base ligands as antileukemia agents. Journal of Molecular Structure, <strong>2024<\/strong>, 1301, art. no. 137400. DOI: 10.1016\/j.molstruc.2023.137400<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Chiacchio, M.A., Campisi, A., Iannazzo, D., <strong>Giofr\u00e8, S.V.<\/strong>, Legnani, L. Design of New Schiff Bases and Their Heavy Metal Ion Complexes for Environmental Applications: A Molecular Dynamics and Density Function Theory Study. <em>International Journal of Molecular Sciences<\/em>, <strong>2024<\/strong>, <em>25<\/em> (8). DOI: 10.3390\/ijms25084159<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Taghizadeh Shool, M., Amiri Rudbari, H., Cuevas-Vicario, J.V., Rodr\u00edguez-Rubio, A., Stagno, C., <strong>Iraci, N.<\/strong>, Efferth, T., Omer, E.A., Schirmeister, T., Blacque, O., Moini, N., Sheibani, E., Micale, N. Investigating the Cytotoxicity of Ru(II) Polypyridyl Complexes by Changing the Electronic Structure of Salicylaldehyde Ligands. Inorganic Chemistry, <strong>2024<\/strong>, <em>63<\/em> (2), pp. 1083-1101. DOI: 10.1021\/acs.inorgchem.3c03414<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Romeo, R., Legnani, L., Chiacchio, M.A., <strong>Giofr\u00e9, S.V.<\/strong>, Iannazzo, D. Antiviral Compounds to Address Influenza Pandemics: An Update from 2016-2022. <em>Current Medicinal Chemistry<\/em>, <strong>2024<\/strong>, 31 (18), 2507-2549. DOI: 10.2174\/0929867331666230907093501<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Iannazzo, D., Celesti, C., <strong>Giofr\u00e8, S.V.<\/strong>, Ettari, R., Bitto, A. Theranostic Applications of 2D Graphene-Based Materials for Solid Tumors Treatment. <em>Nanomaterials<\/em>, <strong>2023<\/strong>, 13 (16), art. no. 2380. DOI: 10.3390\/nano13162380<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Marsili, G., Acchioni, C., Remoli, A.L., Amatore, D., Sgarbanti, R., De Angelis, M., Orsatti, R., Acchioni, M., Astolfi, A., <strong>Iraci, N.<\/strong>, Puzelli, S., Facchini, M., Perrotti, E., Cecchetti, V., Sabatini, S., Superti, F., Agamennone, M., Barreca, M.L., Hiscott, J., Nencioni, L., Sgarbanti, M. Identification of Anti-Influenza A Compounds Inhibiting the Viral Non-Structural Protein 1 (NS1) Using a Type I Interferon-Driven Screening Strategy. <em>International Journal of Molecular Sciences<\/em>, <strong>2023<\/strong>, <em>24<\/em> (13), art. no. 10495. DOI: 10.3390\/ijms241310495<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Iannazzo, D., Giofr\u00e9, S.V. Editorial overview: New synthetic methods: How chemistry change course for a sustainable future. <em>Current Opinion in Green and Sustainable Chemistry<\/em>, <strong>2023<\/strong>, <em>41<\/em>, art. no. 100828. DOI: 10.1016\/j.cogsc.2023.100828<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Smeriglio, A., <strong>Iraci, N.<\/strong>, Denaro, M., Mandalari, G., <strong>Giofr\u00e8, S.V.<\/strong>, Trombetta, D. Synergistic Combination of Citrus Flavanones as Strong Antioxidant and COX-Inhibitor Agent. <em>Antioxidants<\/em>, <strong>2023<\/strong>, <em>12 <\/em>(4), art. no. 972. DOI: 10.3390\/antiox12040972<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">De Gaetano, F., Scala, A., Celesti, C., Lambertsen Larsen, K., Genovese, F., Bongiorno, C., Leggio, L., Iraci, N., <strong>Iraci, N.<\/strong>, Mazzaglia, A., Ventura, C.A. Amphiphilic Cyclodextrin Nanoparticles as Delivery System for Idebenone: A Preformulation Study. <em>Molecules<\/em>, <strong>2023<\/strong>, 28 (7), art. no. 3023. DOI: 10.3390\/molecules28073023<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\"><strong>Giofr\u00e8, S.V.<\/strong>, Celesti, C., Mistretta, G., Tiecco, M. Affinity of deep eutectic solvents with aromatic molecules and aromatic nanostructures in chemical transformations. <em>Current Opinion in Green and Sustainable Chemistry<\/em>, <strong>2023<\/strong>, 40, art. no. 100779. DOI: 10.1016\/j.cogsc.2023.100779<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Di Pietro, M.L., Stagno, C., Efferth, T., Omer, E.A., D\u2019Angelo, V., German\u00f2, M.P., Cacciola, A., De Gaetano, F., <strong>Iraci, N.<\/strong>, Micale, N. Antileukemia Activity and Mechanism of Platinum(II)-Based Metal Complexes. <em>Molecules<\/em>, <strong>2022<\/strong>, 27 (24), art. no. 9000. DOI: 10.3390\/molecules27249000<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Iannazzo, D., Celesti, C., Espro, C., Ferlazzo, A., <strong>Giofr\u00e8, S.V.<\/strong>, Scuderi, M., Scalese, S., Gabriele, B., Mancuso, R., Ziccarelli, I., Visalli, G., Di Pietro, A. Orange-Peel-Derived Nanobiochar for Targeted Cancer Therapy. <em>Pharmaceutics<\/em>, <strong>2022<\/strong>, <em>14<\/em> (10), art. no. 2249. DOI: 10.3390\/pharmaceutics14102249<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Musella, S., Carotenuto, L., <strong>Iraci, N.<\/strong>, Baroli, G., Ciaglia, T., Nappi, P., Basilicata, M.G., Salviati, E., Barrese, V., Vestuto, V., Pignataro, G., Pepe, G., Sommella, E., Di Sarno, V., Manfra, M., Campiglia, P., Gomez-Monterrey, I., Bertamino, A., Taglialatela, M., Ostacolo, C., Miceli, F. Beyond Retigabine: Design, Synthesis, and Pharmacological Characterization of a Potent and Chemically Stable Neuronal Kv7 Channel Activator with Anticonvulsant Activity<em>. <\/em><em>Journal of Medicinal Chemistry<\/em>, <strong>2022<\/strong>, 65 (16), pp. 11340-11364. 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Allosteric inhibition of the hepatitis C virus NS5B polymerase: In silico strategies for drug discovery and development. <em>Future Medicinal Chemistry<\/em>, <strong>2011<\/strong>, 3 (8), pp. 1027-1055. DOI: 10.4155\/fmc.11.53<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Romeo, R., <strong>Giofr\u00e8, S.V.<\/strong>, Iaria, D., Sciortino, M.T., Ronsisvalle, S., Chiacchio, M.A., Scala, A. Synthesis of 5-alkynyl isoxazolidinyl nucleosides. <em>European Journal of Organic Chemistry<\/em>, <strong>2011<\/strong>, (28), 5690-5695. DOI: 10.1002\/ejoc.201100767<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Ettari, R., Zappal\u00e0, M., Micale, N., Grazioso, G., <strong>Giofr\u00e8, S.<\/strong>, Schirmeister, T., Grasso, S. Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors. <em>European Journal of Medicinal Chemistry<\/em>, <strong>2011<\/strong>, <em>46<\/em> (6), 2058-2065. 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Response of a simian immunodeficiency virus (SIVmac251) to raltegravir: A basis for a new treatment for simian AIDS and an animal model for studying lentiviral persistence during antiretroviral therapy. <em>Retrovirology<\/em>, <strong>2010<\/strong>, 7, art. no. 21. DOI: 10.1186\/1742-4690-7-21<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Monforte, A.-M., Logoteta, P., Luca, L.D., <strong>Iraci, N.<\/strong>, Ferro, S., Maga, G., De Clercq, E., Pannecouque, C., Chimirri, A. Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors. <em>Bioorganic and Medicinal Chemistry<\/em>, <strong>2010<\/strong>, 18 (4), pp. 1702-1710. DOI: 10.1016\/j.bmc.2009.12.059<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Piperno, A., <strong>Giofr\u00e8, S.V.<\/strong>, Iannazzo, D., Romeo, R., Romeo, G., Chiacchio, U., Rescifina, A., Piotrowska, D.G. Synthesis of C-4\u2032Truncated Phosphonated Carbocyclic 2\u2032-Oxa-3\u2032-azanucleosides as Antiviral Agents. <em>Journal of Organic Chemistry<\/em>, <strong>2010<\/strong>, <em>75<\/em> (9), 2798-2805. DOI: 10.1021\/jo902485m<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Romeo, G., <strong>Giofr\u00e9, S.V.<\/strong>, Piperno, A., Romeo, R., Chiacchiob, M.A. Synthesis of N,O-homonucleosides with high conformational freedom. Arkivoc, <strong>2009<\/strong> (8), 168-176. DOI: 10.3998\/ark.5550190.0010.814<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Barreca, M.L., <strong>Iraci, N.<\/strong>, De Luca, L., Chimirri, A. Induced-fit docking approach provides insight into the binding mode and mechanism of action of HIV-1 integrase inhibitors. <em>ChemMedChem<\/em>, <strong>2009<\/strong>, 4 (9), pp. 1446-1456. DOI: 10.1002\/cmdc.200900166<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Monforte, A.-M., Logoteta, P., Ferro, S., Luca, L.D., <strong>Iraci, N.<\/strong>, Maga, G., Clercq, E.D., Pannecouque, C., Chimirri, A. Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents. <em>Bioorganic and Medicinal Chemistry<\/em>, <strong>2009<\/strong>, 17 (16), pp. 5962-5967. DOI: 10.1016\/j.bmc.2009.06.068<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">De Luca, L., Barreca, M.L., Ferro, S., Christ, F., <strong>Iraci, N.<\/strong>, Gitto, R., Monforte, A.M., Debyser, Z., Chimirri, A. Pharmacophore-based discovery of small-molecule inhibitors of protein-protein interactions between HIV-1 integrase and cellular cofactor LEDGF\/p75. <em>ChemMedChem<\/em>, <strong>2009<\/strong>, 4 (8), pp. 1311-1316. DOI: 10.1002\/cmdc.200900070<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Ferro, S., De Luca, L., Barreca, M.L., <strong>Iraci, N.<\/strong>, De Grazia, S., Christ, F., Witvrouw, M., Debyser, Z., Chimirri, A. Docking studies on a new human immunodeficiency virus integrase-Mg-DNA complex: phenyl ring exploration and synthesis of 1H-benzylindole derivatives through fluorine substitutions. <em>Journal of medicinal chemistry<\/em>, <strong>2009<\/strong>, 52 (2), pp. 569-573. DOI: 10.1021\/jm8009266<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Stancanelli, R., Crupi, V., De Luca, L., Ficarra, P., Ficarra, R., Gitto, R., Guardo, M., <strong>Iraci, N.<\/strong>, Majolino, D., Tommasini, S., Venuti, V. Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with \u03b2-cyclodextrin. <em>Bioorganic and Medicinal Chemistry<\/em>, <strong>2008<\/strong>, 16 (18), pp. 8706-8712. DOI: 10.1016\/j.bmc.2008.07.085<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Monforte, A.-M., Rao, A., Logoteta, P., Ferro, S., De Luca, L., Barreca, M.L., <strong>Iraci, N.<\/strong>, Maga, G., De Clercq, E., Pannecouque, C., Chimirri, A. Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors. <em>Bioorganic and Medicinal Chemistry<\/em>, <strong>2008<\/strong>, 16 (15), pp. 7429-7435. DOI: 10.1016\/j.bmc.2008.06.012<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">De Luca, L., Barreca, M.L., Ferro, S., <strong>Iraci, N.<\/strong>, Michiels, M., Christ, F., Debyser, Z., Witvrouw, M., Chimirri, A. A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series. <em>Bioorganic and Medicinal Chemistry Letters<\/em>, <strong>2008<\/strong>, 18 (9), pp. 2891-2895. DOI: 10.1016\/j.bmcl.2008.03.089<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Piperno, A., Chiacchio, U., Iannazzo, D., <strong>Giofr\u00e8, S.V.<\/strong>, Romeo, G., Romeo, R. First example of direct RuO4- catalyzed oxidation of isoxazolidines to 3-isoxazolidones. <em>Journal of Organic Chemistry<\/em>, <strong>2007<\/strong>, <em>72<\/em> (10), 3958-3960. DOI: 10.1021\/jo070211n<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Barreca, M.L., Ortuso, F., <strong>Iraci, N.<\/strong>, De Luca, L., Alcaro, S., Chimirri, A. Tn5 transposase as a useful platform to simulate HIV-1 integrase inhibitor binding mode. <em>Biochemical and Biophysical Research Communications<\/em>, <strong>2007<\/strong>, 363 (3), pp. 554-560. DOI: 10.1016\/j.bbrc.2007.08.199<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Barreca, M.L., Rao, A., Luca, L.D., <strong>Iraci, N.<\/strong>, Monforte, A.-M., Maga, G., Clercq, E.D., Pannecouque, C., Balzarini, J., Chimirri, A. Discovery of novel benzimidazolones as potent non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains. <em>Bioorganic and Medicinal Chemistry Letters<\/em>, <strong>2007<\/strong>, 17 (7), pp. 1956-1960. DOI: 10.1016\/j.bmcl.2007.01.025<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Barreca, M.L., De Luca, L., <strong>Iraci, N.<\/strong>, Rao, A., Ferro, S., Maga, G., Chimirri, A. Structure-based pharmacophore identification of new chemical scaffolds as non-nucleoside reverse transcriptase inhibitors. <em>Journal of Chemical Information and Modeling<\/em>, <strong>2007<\/strong>, 47 (2), pp. 557-562. DOI: 10.1021\/ci600320q<\/span><\/li><\/ul>\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-279a72e elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"279a72e\" data-element_type=\"section\" data-e-type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-c807153 elementor-invisible\" data-id=\"c807153\" data-element_type=\"column\" data-e-type=\"column\" data-settings=\"{&quot;background_background&quot;:&quot;classic&quot;,&quot;animation&quot;:&quot;fadeInLeft&quot;}\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-7d47b76 elementor-widget elementor-widget-heading\" data-id=\"7d47b76\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h4 class=\"elementor-heading-title elementor-size-default\"><a href=\"https:\/\/portale.unime.it\/modellopersona\/ricerca\/\">VOLUMI<\/a><\/h4>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-cd9862f elementor-view-default elementor-widget elementor-widget-icon\" data-id=\"cd9862f\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"icon.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<div class=\"elementor-icon-wrapper\">\n\t\t\t<div class=\"elementor-icon\">\n\t\t\t<svg aria-hidden=\"true\" class=\"e-font-icon-svg e-far-newspaper\" viewBox=\"0 0 576 512\" xmlns=\"http:\/\/www.w3.org\/2000\/svg\"><path d=\"M552 64H112c-20.858 0-38.643 13.377-45.248 32H24c-13.255 0-24 10.745-24 24v272c0 30.928 25.072 56 56 56h496c13.255 0 24-10.745 24-24V88c0-13.255-10.745-24-24-24zM48 392V144h16v248c0 4.411-3.589 8-8 8s-8-3.589-8-8zm480 8H111.422c.374-2.614.578-5.283.578-8V112h416v288zM172 280h136c6.627 0 12-5.373 12-12v-96c0-6.627-5.373-12-12-12H172c-6.627 0-12 5.373-12 12v96c0 6.627 5.373 12 12 12zm28-80h80v40h-80v-40zm-40 140v-24c0-6.627 5.373-12 12-12h136c6.627 0 12 5.373 12 12v24c0 6.627-5.373 12-12 12H172c-6.627 0-12-5.373-12-12zm192 0v-24c0-6.627 5.373-12 12-12h104c6.627 0 12 5.373 12 12v24c0 6.627-5.373 12-12 12H364c-6.627 0-12-5.373-12-12zm0-144v-24c0-6.627 5.373-12 12-12h104c6.627 0 12 5.373 12 12v24c0 6.627-5.373 12-12 12H364c-6.627 0-12-5.373-12-12zm0 72v-24c0-6.627 5.373-12 12-12h104c6.627 0 12 5.373 12 12v24c0 6.627-5.373 12-12 12H364c-6.627 0-12-5.373-12-12z\"><\/path><\/svg>\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-f472f9a\" data-id=\"f472f9a\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-053a327 elementor-widget elementor-widget-text-editor\" data-id=\"053a327\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t\t\t<p><span style=\"color: #333333\"><span style=\"font-family: tahoma, arial, helvetica, sans-serif;font-size: 10pt\"><strong style=\"background-color: var(--global--color-background)\"><u><strong>VOLUMI<\/strong><\/u><\/strong><\/span><\/span><\/p><ul><li><span style=\"font-size: 10pt;color: #000000\">Chemical Synthesis of Nucleoside Analogues. Pedro Merino (editor) ISBN: 978-1-1180-0751-8. Ugo Chiacchio, Antonio Corsaro, <strong>Salvatore Giofr\u00e8<\/strong>, Giovanni Romeo. <em>Isoxazolidinyl Nucleosides.<\/em> Cap. 17, pp 781-818. <strong>2013. <\/strong>ISBN: 978-1-118-00751-8.<\/span><\/li><li><span style=\"font-size: 10pt;color: #000000\">Therapy of Viral Infections. Topics in Medicinal Chemistry. Wibke E. Diederich, Holger Steuber. Springer Berlin-Heidelberg<strong><em>.<\/em><\/strong> Beatrice Macchi,\u00a0Giovanni Romeo,\u00a0Ugo Chiacchio, Caterina Frezza, <strong>Salvatore V. Giofr\u00e8<\/strong>,<strong>\u00a0<\/strong>Francesca Marino-Merlo. <em>Phosphonated Nucleoside Analogues as Antiviral Agents<\/em>. Volume 15,\u00a0<strong>2015<\/strong>,\u00a053-91. Print ISBN:978-3-662-46758-9. Online ISBN:978-3-662-46759-6.<\/span><\/li><\/ul>\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-bdf3fba elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"bdf3fba\" data-element_type=\"section\" data-e-type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-7b9af6a elementor-invisible\" data-id=\"7b9af6a\" data-element_type=\"column\" data-e-type=\"column\" data-settings=\"{&quot;background_background&quot;:&quot;classic&quot;,&quot;animation&quot;:&quot;fadeInLeft&quot;}\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-51fc9dd elementor-widget elementor-widget-heading\" data-id=\"51fc9dd\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"heading.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<h4 class=\"elementor-heading-title elementor-size-default\"><a href=\"https:\/\/portale.unime.it\/modellopersona\/ricerca\/\">BREVETTI<\/a><\/h4>\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-404c7cd elementor-view-default elementor-widget elementor-widget-icon\" data-id=\"404c7cd\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"icon.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<div class=\"elementor-icon-wrapper\">\n\t\t\t<div class=\"elementor-icon\">\n\t\t\t<svg aria-hidden=\"true\" class=\"e-font-icon-svg e-fas-book\" viewBox=\"0 0 448 512\" xmlns=\"http:\/\/www.w3.org\/2000\/svg\"><path d=\"M448 360V24c0-13.3-10.7-24-24-24H96C43 0 0 43 0 96v320c0 53 43 96 96 96h328c13.3 0 24-10.7 24-24v-16c0-7.5-3.5-14.3-8.9-18.7-4.2-15.4-4.2-59.3 0-74.7 5.4-4.3 8.9-11.1 8.9-18.6zM128 134c0-3.3 2.7-6 6-6h212c3.3 0 6 2.7 6 6v20c0 3.3-2.7 6-6 6H134c-3.3 0-6-2.7-6-6v-20zm0 64c0-3.3 2.7-6 6-6h212c3.3 0 6 2.7 6 6v20c0 3.3-2.7 6-6 6H134c-3.3 0-6-2.7-6-6v-20zm253.4 250H96c-17.7 0-32-14.3-32-32 0-17.6 14.4-32 32-32h285.4c-1.9 17.1-1.9 46.9 0 64z\"><\/path><\/svg>\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-4a35824\" data-id=\"4a35824\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-5234c27 elementor-widget elementor-widget-text-editor\" data-id=\"5234c27\" data-element_type=\"widget\" data-e-type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t\t\t<p><span style=\"color: #333333\"><span style=\"font-family: tahoma, arial, helvetica, sans-serif;font-size: 10pt\"><strong style=\"background-color: var(--global--color-background)\"><u>BREVETTI<\/u><\/strong><\/span><\/span><\/p>\n<ul>\n<li><span style=\"font-size: 10pt;color: #000000\">Uso di Derivati 2-Oxo-2H-Pirrol-1(5<em>H<\/em>)-Carbossamidici come Agenti Anti-HIV e Processo per la loro Produzione. <strong>Depositato il 4-03-2016, numero 102016000022765 (UA2016A001346), <\/strong>data di pubblicazione 05-09-2017, Concesso il 14-09-2018.<\/span><\/li>\n<li><span style=\"font-size: 10pt;color: #000000\"><span style=\"font-size: 10pt\">Prion protein ligands as therapeutic agents for neurodegenerative disorders. <strong>Depositato il 06-08-2013 numero 10391068 (<\/strong><\/span><strong>US10391068B2),<\/strong> data di pubblicazione 16-07-2015 (<a id=\"link\" class=\"style-scope state-modifier\" style=\"color: #000000\" href=\"https:\/\/patents.google.com\/patent\/US20150196508A1\/en?peid=62f0942d1cda8%3A85%3A929f236c\"><span class=\"title-text style-scope application-timeline\">US20150196508A1<\/span><\/a>), concesso il 27-08-2019 (<a id=\"link\" class=\"style-scope state-modifier\" href=\"https:\/\/patents.google.com\/patent\/US10391068B2\/en?peid=62f094908f598%3A90%3A169de58c\"><span class=\"title-text style-scope application-timeline\">US10391068B2<\/span><\/a>).<\/span><\/li>\n<li><span style=\"font-size: 10pt;color: #000000\">Novel potassium channel inhibitors. <strong>Depositato il 21-09-2021 numero PCT\/EP2021\/075923<\/strong>, data di pubblicazione 31-03-2022 (<a id=\"link\" class=\"style-scope state-modifier\" style=\"color: #000000\" href=\"https:\/\/patents.google.com\/patent\/WO2022063767A1\/en?peid=62f099fa239a0%3Ac0%3A86465be0\"><span class=\"title-text style-scope application-timeline\">WO2022063767A1<\/span><\/a>).<\/span><span style=\"font-size: 10pt;color: #000000\">&nbsp;<\/span><\/li>\n<\/ul>\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section class=\"elementor-section elementor-top-section elementor-element elementor-element-e387566 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"e387566\" data-element_type=\"section\" data-e-type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-97f572d\" data-id=\"97f572d\" data-element_type=\"column\" data-e-type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap\">\n\t\t\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<\/div>\n\t\t","protected":false},"excerpt":{"rendered":"<p>PUBBLICAZIONI LE PUBBLICAZIONI Il gruppo di ricerca DESY LAB pubblica articoli su riviste scientifiche di interesse internazionale Topics: Graphene; Quantum Dot; Biocompatibility; Heavy Metal; Bioaccumulation; Environmental Monitoring; Nitrone; Heterocyclic Compound; Stereoselective Synthesis; Citrus; Flavonoid; Antioxidant Capacity; Antivirus Agent; Nanoparticle; COVID-19; Potassium Channel; Retigabine; Encephalopathy; Transient Receptor Potential Channel; Ankyrin; Sensory Receptor Cell; Human Immunodeficiency Virus&hellip; <a class=\"more-link\" href=\"https:\/\/portale2.unime.it\/desylab\/pubblicazioni\/\">Continua a leggere <span class=\"screen-reader-text\">PUBBLICAZIONI<\/span><\/a><\/p>\n","protected":false},"author":1,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"elementor_header_footer","meta":{"footnotes":""},"class_list":["post-1372","page","type-page","status-publish","hentry","entry"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ 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